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| New compound sets identified from high throughput phenotypic screening against three kinetoplastid parasites: an open resource I Pena, M Pilar Manzano, J Cantizani, A Kessler, J Alonso-Padilla, ... Scientific reports 5 (1), 8771, 2015 | 269 | 2015 |
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| Quantitative, wide-spectrum kinase profiling in live cells for assessing the effect of cellular ATP on target engagement JD Vasta, CR Corona, J Wilkinson, CA Zimprich, JR Hartnett, MR Ingold, ... Cell chemical biology 25 (2), 206-214. e11, 2018 | 212 | 2018 |
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| Discovery and characterization of GSK2801, a selective chemical probe for the bromodomains BAZ2A and BAZ2B P Chen, A Chaikuad, P Bamborough, M Bantscheff, C Bountra, C Chung, ... Journal of medicinal chemistry 59 (4), 1410-1424, 2016 | 159 | 2016 |
| Progress towards a public chemogenomic set for protein kinases and a call for contributions DH Drewry, CI Wells, DM Andrews, R Angell, H Al-Ali, AD Axtman, ... PloS one 12 (8), e0181585, 2017 | 150 | 2017 |
| Discovery of GSK1070916, a potent and selective inhibitor of Aurora B/C kinase ND Adams, JL Adams, JL Burgess, AM Chaudhari, RA Copeland, ... Journal of medicinal chemistry 53 (10), 3973-4001, 2010 | 125 | 2010 |
| Seeding collaborations to advance kinase science with the GSK Published Kinase Inhibitor Set (PKIS) D H Drewry, T M Willson, W J Zuercher Current topics in medicinal chemistry 14 (3), 340-342, 2014 | 124 | 2014 |
| Plasmodium kinases as targets for new-generation antimalarials IS Lucet, A Tobin, D Drewry, AF Wilks, C Doerig Future medicinal chemistry 4 (18), 2295-2310, 2012 | 100 | 2012 |
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| The kinase chemogenomic set (KCGS): an open science resource for kinase vulnerability identification CI Wells, H Al-Ali, DM Andrews, CRM Asquith, AD Axtman, I Dikic, ... International journal of molecular sciences 22 (2), 566, 2021 | 79 | 2021 |
| Profile of the GSK published protein kinase inhibitor set across ATP-dependent and-independent luciferases: implications for reporter-gene assays P Dranchak, R MacArthur, R Guha, WJ Zuercher, DH Drewry, DS Auld, ... PloS one 8 (3), e57888, 2013 | 78 | 2013 |
